Reference Library

Peptide Encyclopedia

Research-grade reference on 444 compounds: published dose and cycle ranges, safety profiles, evidence quality, and common misconceptions. ProtoComp guidance is grounded in published research. Always confirm with your clinician before changing your protocol.

444 compounds

1-Androstenediol

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

1-Androstenedione

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

1-Androsterone

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

1-Testosterone

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

11-Ketodihydrotestosterone

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

11-Ketotestosterone

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

19-Nor-5-androstenediol

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

19-Nor-5-androstenedione

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

19-Nordehydroepiandrosterone

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

4-androstene-3,6,17-trione

Metabolic

Metabolic reference profile.

preclinical only

4-Androstenediol

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

4-Dehydroepiandrosterone

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

4-Hydroxytestosterone

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

5-Amino-1MQ

Metabolic

Metabolic reference profile.

preclinical only

5-Androstenedione

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

6-isoquinoline-1-carbonitrile

SARM

SARM reference profile.

preclinical only· WADA banned

7,8-DHF

Nootropic

Nootropic reference profile.

preclinical only

7,8-Dihydroxyflavone

Metabolic

Metabolic reference profile.

preclinical only

9-Me-BC

Nootropic

Nootropic reference profile.

preclinical only

Abarelix

Healing

Healing reference profile.

limited human data

AC-262536

SARM

SARM reference profile.

preclinical only· WADA banned

acacetin

Metabolic

Metabolic reference profile.

preclinical only

Acarbose

Metabolic

Metabolic reference profile.

preclinical only

ACE-031

Healing

Healing reference profile.

preclinical only

ACE-083

Healing

Healing reference profile.

preclinical only

Acetyl-L-Carnitine

Metabolic

Metabolic reference profile.

preclinical only

ACP-105

SARM

SARM reference profile.

preclinical only· WADA banned

Acyline

Healing

Healing reference profile.

preclinical only

Adamax

Nootropic

Nootropic reference profile.

preclinical only

Adrenosterone

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Afamelanotide

Healing

Healing reference profile.

limited human data

Albuterol

Fat Loss

Fat Loss reference profile.

preclinical only· WADA banned

Alirocumab

Metabolic

Metabolic reference profile.

preclinical only

Alpha-GPC

Nootropic

Nootropic reference profile.

preclinical only

Aminoglutethimide

Metabolic

Metabolic reference profile.

preclinical only

Amitriptyline

Metabolic

Metabolic reference profile.

preclinical only

Amycretin

Metabolic

Metabolic reference profile.

limited human data

Anamorelin

GH Secretagogue

GH Secretagogue reference profile.

preclinical only

Anastrozole

Metabolic

Metabolic reference profile.

preclinical only

Andarine

SARM

SARM reference profile.

preclinical only· WADA banned

Androisoxazole

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

androsta-1,4,6-triene-3,17-dione

Metabolic

Metabolic reference profile.

preclinical only

Androstenediol

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Androstenedione

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Androsterone

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

AOD-9604

Fat Loss

Beyond 500 mcg/day shows no additional benefit. Morning preferred.

limited human data· WADA banned

apigenin

Metabolic

Metabolic reference profile.

preclinical only

Arformoterol

Fat Loss

Fat Loss reference profile.

preclinical only· WADA banned

Ashwagandha

Metabolic

Metabolic reference profile.

preclinical only

Atamestane

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Azagly-nafarelin

Healing

Healing reference profile.

preclinical only

Azaline B

Healing

Healing reference profile.

preclinical only

baicalein

Metabolic

Metabolic reference profile.

preclinical only

Bambuterol

Fat Loss

Fat Loss reference profile.

preclinical only· WADA banned

bazedoxifene

Metabolic

Metabolic reference profile.

preclinical only

bazedoxifene acetate

Metabolic

Metabolic reference profile.

preclinical only

BCAAs

Metabolic

Metabolic reference profile.

preclinical only

BDNF Peptides

Nootropic

Nootropic reference profile.

preclinical only

Beetroot Extract

Metabolic

Metabolic reference profile.

preclinical only

Berberine

Metabolic

Metabolic reference profile.

preclinical only

Beta-Alanine

Metabolic

Metabolic reference profile.

preclinical only

Betaine Anhydrous

Metabolic

Metabolic reference profile.

preclinical only

bifonazole

Metabolic

Metabolic reference profile.

preclinical only

Bimagrumab

Metabolic

Metabolic reference profile.

preclinical only

biochanin A

Metabolic

Metabolic reference profile.

preclinical only

Bitolterol

Fat Loss

Fat Loss reference profile.

preclinical only· WADA banned

BMS-564929

SARM

SARM reference profile.

preclinical only· WADA banned

Bolandiol

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Bolandione

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Bolasterone

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Bolazine

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Boldenone

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Boldenone Undecylenate

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Boldione

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Bolenol

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Bolmantalate

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Boron

Metabolic

Metabolic reference profile.

preclinical only

BPC-157

Healing

Split AM/PM for stable blood levels. Oral dose higher (500-1000 mcg/day) for gut-specific use.

limited human data· WADA banned

Bremelanotide

Healing

Healing reference profile.

limited human data

Buserelin

Healing

Healing reference profile.

preclinical only

Caffeine

Fat Loss

Fat Loss reference profile.

preclinical only· WADA banned

Cagrilintide

Metabolic

Long-acting amylin analog. Investigational — Phase 3 trials ongoing, often co-administered with Semaglutide (CagriSema). Dose range refle…

limited human data

CagriSema

Metabolic

Metabolic reference profile.

limited human data

Calusterone

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Capromorelin

GH Secretagogue

GH Secretagogue reference profile.

preclinical only

Cardarine

SARM

SARM reference profile.

preclinical only· WADA banned

Cerebrolysin

Nootropic

Porcine-derived peptide preparation. Approved in many European and Asian countries for stroke, TBI, and dementia. Dose is in mL of a stan…

strong human data

Cetrorelix

Healing

Healing reference profile.

limited human data

Chlorodehydromethylandrostenediol

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Chlorodehydromethyltestosterone

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Chloromethylandrostenediol

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

chrysin

Metabolic

Metabolic reference profile.

preclinical only

Citicoline

Nootropic

Nootropic reference profile.

preclinical only

Citrulline Malate

Metabolic

Metabolic reference profile.

preclinical only

CJC-1293

Healing

Healing reference profile.

preclinical only

CJC-1295

GH Secretagogue

GH Secretagogue reference profile.

preclinical only

CJC-1295

GH Secretagogue

Short-acting. Half-life ~30 min. Multiple daily doses needed.

limited human data· WADA banned

CJC-1295 (with DAC)

GH Secretagogue

2 mg SubQ 1-2x/week. Some sources say 2-3 mg/week. Half-life 5.8-8.1 days.

limited human data· WADA banned

CJC-1295 DAC

GH Secretagogue

GH Secretagogue reference profile.

preclinical only

CJC-1295 No DAC

GH Secretagogue

GH Secretagogue reference profile.

preclinical only

Clenbuterol

Fat Loss

Fat Loss reference profile.

preclinical only· WADA banned

Clomiphene

Metabolic

Metabolic reference profile.

preclinical only

Clostebol

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

clotrimazole

Metabolic

Metabolic reference profile.

preclinical only

Cloxotestosterone

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Collagen Peptides

Metabolic

Metabolic reference profile.

preclinical only

CoQ10

Metabolic

Metabolic reference profile.

preclinical only

Cortagen

Healing

Healing reference profile.

preclinical only

Cotadutide

Metabolic

Metabolic reference profile.

limited human data

coumestrol

Metabolic

Metabolic reference profile.

preclinical only

Creatine HCl

Metabolic

Metabolic reference profile.

preclinical only

Creatine Monohydrate

Metabolic

Metabolic reference profile.

preclinical only

Danazol

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Danuglipron

Metabolic

Metabolic reference profile.

limited human data

Degarelix

Healing

Healing reference profile.

limited human data

Dehydroandrosterone

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Dehydroepiandrosterone

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Deslorelin

Healing

Healing reference profile.

preclinical only

Desoxymethyltestosterone

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

DHEA

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

DHT Gel

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Dianabol

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Dienedione

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Dienolone

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Dihexa

Nootropic

Nootropic reference profile.

preclinical only

Dihydrotestosterone

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Dimethandrolone

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Dimethyldienolone

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Dimethyltrienolone

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

DNP

Fat Loss

Fat Loss reference profile.

preclinical only· WADA banned

Drostanolone

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Drostanolone Enanthate

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Drostanolone Propionate

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

DSIP

Nootropic

Short half-life peptide with sleep-modulating effects. Most human data is from older Russian literature.

limited human data

Dulaglutide

Metabolic

FDA-approved weekly GLP-1 RA for T2D. Titrate 0.75 then 1.5 then 3 then 4.5 mg weekly, at least 4 weeks between steps.

strong human data

EAAs

Metabolic

Metabolic reference profile.

preclinical only

Efinopegdutide

Metabolic

Metabolic reference profile.

limited human data

Elagolix

Healing

Healing reference profile.

preclinical only

Electrolytes

Metabolic

Metabolic reference profile.

preclinical only

Eloralintide

Metabolic

Metabolic reference profile.

limited human data

Enclomiphene

Metabolic

Metabolic reference profile.

preclinical only

Enestebol

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

enilconazole

Metabolic

Metabolic reference profile.

preclinical only

Enobosarm

SARM

SARM reference profile.

preclinical only· WADA banned

Ephedrine

Fat Loss

Fat Loss reference profile.

preclinical only· WADA banned

Epiandrosterone

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

epigallocatechin gallate

Metabolic

Metabolic reference profile.

preclinical only

Epitalon

Anti-Aging

Anti-Aging reference profile.

animal only

Epithalon

Healing

Healing reference profile.

preclinical only

Epitiostanol

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Ethisterone

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Ethyldienolone

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Ethylestrenol

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Ethyltestosterone

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Etynodiol

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Evolocumab

Metabolic

Metabolic reference profile.

preclinical only

Exemestane

Metabolic

Metabolic reference profile.

preclinical only

Exenatide

Metabolic

Metabolic reference profile.

limited human data

Exenatide ER

Metabolic

Metabolic reference profile.

limited human data

Ezetimibe

Metabolic

Metabolic reference profile.

preclinical only

Fadrozole

Metabolic

Metabolic reference profile.

preclinical only

Fenoterol

Fat Loss

Fat Loss reference profile.

preclinical only· WADA banned

Fertirelin

Healing

Healing reference profile.

preclinical only

Fluoxymesterone

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Follistatin 315

Healing

Healing reference profile.

preclinical only

Follistatin 344

Growth Factor

No published human trials. Dosing is extrapolated from animal data and anecdotal use.

preclinical only· WADA banned

Follitropin Alfa

Metabolic

Metabolic reference profile.

preclinical only

Follitropin Beta

Metabolic

Metabolic reference profile.

preclinical only

Formebolone

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Formestane

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Formoterol

Fat Loss

Fat Loss reference profile.

preclinical only· WADA banned

FOXO4-DRI

Healing

Healing reference profile.

preclinical only

fulvestrant

Metabolic

Metabolic reference profile.

preclinical only

Furazabol

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Ganirelix

Healing

Healing reference profile.

limited human data

Genotropin

Healing

Healing reference profile.

preclinical only

Gestrinone

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

GHK

Healing

Healing reference profile.

preclinical only

GHK-Cu

Healing

8-12 weeks skin, 12-16 weeks hair (topical)

limited human data

Ghrelin

GH Secretagogue

GH Secretagogue reference profile.

preclinical only

GHRP-1

GH Secretagogue

GH Secretagogue reference profile.

preclinical only

GHRP-2

GH Secretagogue

8-12 weeks. Lower-frequency maintenance possible.

limited human data· WADA banned

GHRP-6

GH Secretagogue

Potent ghrelin mimetic with strong appetite stimulation. Pulses better than higher single doses.

limited human data· WADA banned

Gonadorelin

GH Secretagogue

Synthetic GnRH. FDA-approved (Factrel) for diagnostic LH/FSH evaluation. Used off-label in TRT protocols and post-cycle therapy to mainta…

strong human data

Goserelin

Healing

Healing reference profile.

limited human data

GRF 1-29

Healing

Healing reference profile.

preclinical only

GSK-4336A

SARM

SARM reference profile.

preclinical only· WADA banned

GSK2881078

SARM

SARM reference profile.

preclinical only· WADA banned

GW-501516

SARM

PPAR-δ agonist (not a true SARM). Development was halted after long-term animal studies showed accelerated tumor formation across multipl…

preclinical only· WADA banned

GW0742

SARM

SARM reference profile.

preclinical only· WADA banned

GW590735

SARM

SARM reference profile.

preclinical only· WADA banned

Halotestin

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

hCG

Metabolic

Metabolic reference profile.

preclinical only

Hexarelin

GH Secretagogue

Most potent GHRP per microgram. Rapid receptor desensitization — short cycles only.

limited human data· WADA banned

HGH Fragment 176-191

Fat Loss

C-terminal fragment of hGH. Claimed fat-loss action without the GH/IGF-1 anabolic effects. Most human dosing is anecdotal.

limited human data· WADA banned

Histrelin

Healing

Healing reference profile.

limited human data

HMB

Metabolic

Metabolic reference profile.

preclinical only

HMG

Metabolic

Metabolic reference profile.

preclinical only

Humanin

Healing

Healing reference profile.

preclinical only

Humatrope

Healing

Healing reference profile.

preclinical only

Humulin R

Metabolic

Metabolic reference profile.

limited human data

Hydroxystenozole

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Ibutamoren

GH Secretagogue

GH Secretagogue reference profile.

preclinical only

IGF-1

Healing

Healing reference profile.

preclinical only

IGF-1 DES

Healing

Healing reference profile.

preclinical only

IGF-1 LR3

Growth Factor

Beginners 20-40 mcg. Female athletes 20-40 mcg. 5 days on / 2 off common.

limited human data· WADA banned

IGF-DES

Growth Factor

Post-workout only, injected into trained muscle.

limited human data· WADA banned

Indacaterol

Fat Loss

Fat Loss reference profile.

preclinical only· WADA banned

Insulin Aspart

Metabolic

Metabolic reference profile.

limited human data

Insulin Degludec

Metabolic

Metabolic reference profile.

limited human data

Insulin Detemir

Metabolic

Metabolic reference profile.

limited human data

Insulin Glargine

Metabolic

Metabolic reference profile.

limited human data

Insulin Glulisine

Metabolic

Metabolic reference profile.

limited human data

Insulin Lispro

Metabolic

Metabolic reference profile.

limited human data

Insulin NPH

Metabolic

Metabolic reference profile.

limited human data

Insulin Regular

Metabolic

Metabolic reference profile.

limited human data

Ipamorelin

GH Secretagogue

Bell-shaped dose-response — more is not better. Split into 1-3 doses.

limited human data· WADA banned

Iturelix

Healing

Healing reference profile.

preclinical only

JNJ-28330835

SARM

SARM reference profile.

preclinical only· WADA banned

Ketoconazole Shampoo

Metabolic

Metabolic reference profile.

preclinical only

Kisspeptin-10

Healing

Healing reference profile.

preclinical only

Kisspeptin-54

Healing

Healing reference profile.

preclinical only

KPV

Anti-Inflammatory

Experimental. Animal studies used 1-5 mg/kg.

animal only

L-Arginine

Metabolic

Metabolic reference profile.

preclinical only

L-Citrulline

Metabolic

Metabolic reference profile.

preclinical only

L-Theanine

Nootropic

Nootropic reference profile.

preclinical only

Lanreotide

Healing

Healing reference profile.

limited human data

Larazotide

Healing

Healing reference profile.

limited human data

Lecirelin

Healing

Healing reference profile.

preclinical only

Letrozole

Metabolic

Metabolic reference profile.

preclinical only

Leuprorelin

Healing

Healing reference profile.

preclinical only

Levalbuterol

Fat Loss

Fat Loss reference profile.

preclinical only· WADA banned

Levothyroxine

Metabolic

Metabolic reference profile.

limited human data

LGD-2226

SARM

SARM reference profile.

preclinical only· WADA banned

LGD-3303

SARM

SARM reference profile.

preclinical only· WADA banned

LGD-4033

SARM

Phase 2 trials completed for muscle wasting. Dose-dependent lean mass gain and HPG suppression documented in healthy men at 1 mg/day.

limited human data· WADA banned

Linzagolix

Healing

Healing reference profile.

preclinical only

Liothyronine

Metabolic

Metabolic reference profile.

limited human data

Liraglutide

Metabolic

FDA-approved daily GLP-1 RA. Saxenda (obesity): titrate to 3 mg daily. Victoza (T2D): 0.6-1.8 mg daily.

strong human data

Lixisenatide

Metabolic

Metabolic reference profile.

limited human data

LL-37

Healing

Healing reference profile.

preclinical only

Lotiglipron

Metabolic

Metabolic reference profile.

limited human data

LY 117018

Metabolic

Metabolic reference profile.

preclinical only

Lynestrenol

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Macimorelin

GH Secretagogue

GH Secretagogue reference profile.

preclinical only

Magnesium Glycinate

Metabolic

Metabolic reference profile.

preclinical only

MariTide

Metabolic

Metabolic reference profile.

limited human data

Mazdutide

Fat Loss

Phase 3 GLORY-1 trial in Chinese adults with obesity used 6 mg or 9 mg weekly. Dose-escalation over 4-week intervals.

strong human data

Mebolazine

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Mecasermin

Healing

Healing reference profile.

preclinical only

Melanotan I

Healing

Healing reference profile.

preclinical only

Melanotan II

Nootropic

Non-selective melanocortin receptor agonist. Research chemical — not approved for human use. Loading phase: low daily dose with gradual i…

limited human data

Menotropins

Metabolic

Metabolic reference profile.

preclinical only

MENT

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Mepitiostane

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Mesabolone

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Mestanolone

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Mesterolone

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Metandienone

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Metenolone

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Metenolone Acetate

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Metenolone Enanthate

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Metformin

Metabolic

Metabolic reference profile.

limited human data

Metformin ER

Metabolic

Metabolic reference profile.

limited human data

Methandienone

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Methandriol

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Methasterone

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Methenolone Acetate

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Methenolone Enanthate

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Methoxydienone

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Methyl-1-testosterone

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Methylclostebol

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Methyldiazinol

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Methyldienolone

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Methylepitiostanol

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Methylhydroxynandrolone

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Methylstenbolone

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Methyltestosterone

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Methyltestosterone 3-hexyl ether

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Metribolone

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

MGF

Growth Factor

No published human dosing trials. The endogenous splice variant exists in human muscle, but synthetic MGF protocols are not supported by peer-reviewed dose-finding data.

animal only· WADA banned

Mibolerone

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Minoxidil Topical

Metabolic

Metabolic reference profile.

preclinical only

Mirtazapine

Metabolic

Metabolic reference profile.

preclinical only

MK-0773

SARM

SARM reference profile.

preclinical only· WADA banned

MK-2866

SARM

Most studied SARM in clinical trials — Phase 2 data for muscle wasting, cachexia, and sarcopenia. Dose-dependent HPG effects are milder t…

limited human data· WADA banned

MK-677 (Ibutamoren)

GH Secretagogue

Oral — no injections needed. Once daily.

strong human data· WADA banned

Mod GRF 1-29

Healing

Healing reference profile.

preclinical only

MOTS-c

Metabolic

Mitochondrial-derived peptide. Limited human trials — dosing based on early clinical research.

limited human data

Myostatin Propeptide

Healing

Healing reference profile.

preclinical only

N-Acetyl Semax Amidate

Nootropic

Nootropic reference profile.

preclinical only

NA-Selank Amidate

Nootropic

Nootropic reference profile.

preclinical only

NAC

Metabolic

Metabolic reference profile.

preclinical only

Nafarelin

Healing

Healing reference profile.

limited human data

Nandrolone

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Nandrolone Decanoate

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

nandrolone p-hexyloxyphenylpropionate

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Nandrolone Phenylpropionate

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

NAP

Nootropic

Nootropic reference profile.

preclinical only

Nisterime

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Noopept

Nootropic

Nootropic reference profile.

preclinical only

Norboletone

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Norclostebol

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Norditropin

Healing

Healing reference profile.

preclinical only

Norethandrolone

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Norethisterone

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Norgestrel

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Norgestrienone

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Normethandrone

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Nortriptyline

Metabolic

Metabolic reference profile.

preclinical only

Norvinisterone

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Novarel

Metabolic

Metabolic reference profile.

preclinical only

Novolin R

Metabolic

Metabolic reference profile.

limited human data

Octreotide

Healing

Healing reference profile.

limited human data

Olodaterol

Fat Loss

Fat Loss reference profile.

preclinical only· WADA banned

Omega-3

Metabolic

Metabolic reference profile.

preclinical only

Omnitrope

Healing

Healing reference profile.

preclinical only

OPK-88004

SARM

SARM reference profile.

preclinical only· WADA banned

Oral Minoxidil

Metabolic

Metabolic reference profile.

preclinical only

Orforglipron

Fat Loss

Phase 3 ATTAIN-1 obesity trial uses dose-escalation up to 36 mg daily. Oral, non-peptide structure unlike injectable GLP-1 analogs.

limited human data

Ornirelix

Healing

Healing reference profile.

preclinical only

ospemifene

Metabolic

Metabolic reference profile.

preclinical only

Ostarine

SARM

SARM reference profile.

preclinical only· WADA banned

Oxabolone

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Oxandrolone

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Oxymesterone

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Oxymetholone

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Ozarelix

Healing

Healing reference profile.

preclinical only

P21

Nootropic

Nootropic reference profile.

preclinical only

Pasireotide

Healing

Healing reference profile.

limited human data

PE-22-28

Nootropic

Nootropic reference profile.

animal only

Peforelin

Healing

Healing reference profile.

preclinical only

PEG-MGF

Healing

Healing reference profile.

preclinical only

Pemvidutide

Fat Loss

Phase 2 MOMENTUM (obesity) and IMPACT (MASH) trials used 1.2, 1.8, and 2.4 mg weekly. Phase 3 not yet initiated as of 2026.

limited human data

Penmesterol

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Pinealon

Healing

Healing reference profile.

preclinical only

Pirbuterol

Fat Loss

Fat Loss reference profile.

preclinical only· WADA banned

Plomestane

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

PNC-27

Healing

Healing reference profile.

preclinical only

Pregnenolone

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Pregnyl

Metabolic

Metabolic reference profile.

preclinical only

Procaterol

Fat Loss

Fat Loss reference profile.

preclinical only· WADA banned

Propetandrol

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Prostanozol

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Proviron

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

PT-141

Nootropic

FDA-approved as Vyleesi for HSDD in premenopausal women. Dose as-needed, ≥45 min before anticipated sexual activity. Max 1 dose per 24 ho…

strong human data

Quinbolone

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Quingestanol

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

RAD-140

SARM

Selective androgen receptor modulator. Originally investigated for muscle wasting. Phase 1 trials completed. Research chemical — not appr…

limited human data· WADA banned

RAD-150

SARM

SARM reference profile.

preclinical only· WADA banned

Raloxifene

Metabolic

Metabolic reference profile.

preclinical only

raloxifene hydrochloride

Metabolic

Metabolic reference profile.

preclinical only

Recombinant FSH

Metabolic

Metabolic reference profile.

preclinical only

Relugolix

Healing

Healing reference profile.

preclinical only

Retatrutide

Metabolic

Investigational triple agonist (GLP-1/GIP/glucagon). Phase 3 trials ongoing. Dose range reflects published trial protocols, not FDA-appro…

limited human data

rhGH

Healing

Healing reference profile.

preclinical only

Rhodiola Rosea

Metabolic

Metabolic reference profile.

preclinical only

Ritodrine

Fat Loss

Fat Loss reference profile.

preclinical only· WADA banned

RU-2309

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Rybelsus

Metabolic

Metabolic reference profile.

limited human data

S-101479

SARM

SARM reference profile.

preclinical only· WADA banned

S-23

SARM

Highly potent and suppressive SARM. Investigated as a male contraceptive in preclinical studies due to profound HPG axis suppression.

preclinical only· WADA banned

S-4

SARM

Early SARM investigated for BPH and muscle wasting. Known for dose-dependent yellow vision tint caused by accumulation in retinal tissue.

limited human data· WADA banned

S-40503

SARM

SARM reference profile.

preclinical only· WADA banned

Salbutamol

Fat Loss

Fat Loss reference profile.

preclinical only· WADA banned

Salmeterol

Fat Loss

Fat Loss reference profile.

preclinical only· WADA banned

SARM S1

SARM

SARM reference profile.

preclinical only· WADA banned

Selank

Nootropic

Nootropic reference profile.

limited human data

Semaglutide

Metabolic

FDA-approved GLP-1 RA. Wegovy (obesity): titrate to 2.4 mg weekly. Ozempic (T2D): 0.5-2 mg weekly. Start at 0.25 mg weekly and titrate ev…

strong human data

Semaglutide Oral

Metabolic

Metabolic reference profile.

limited human data

Semax

Nootropic

Split 2-3 doses. Microdosing: 100-200 mcg 1-3x/day.

limited human data

Sermorelin

GH Secretagogue

Once daily pre-bed. Not a quick-fix compound — requires weeks for meaningful results.

limited human data

Setmelanotide

Healing

Healing reference profile.

limited human data

Silandrone

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

SLU-PP

Metabolic

Metabolic reference profile.

preclinical only

SLU-PP-332

SARM

SARM reference profile.

preclinical only· WADA banned

Sodium Bicarbonate

Metabolic

Metabolic reference profile.

preclinical only

Somatostatin

Healing

Healing reference profile.

preclinical only

Somatropin

Healing

Healing reference profile.

preclinical only

SR9009

SARM

REV-ERB agonist (not a true SARM). Poor oral bioavailability — the compound sold to users as SR9009 likely has very limited systemic effe…

preclinical only· WADA banned

SR9011

SARM

SARM reference profile.

preclinical only· WADA banned

SS-20

Healing

Healing reference profile.

preclinical only

SS-31

Anti-Aging

Anti-Aging reference profile.

limited human data

Stanozolol

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Stanozolol Injectable

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Stanozolol Oral

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Stenabolic

SARM

SARM reference profile.

preclinical only· WADA banned

Stenbolone

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Superdrol

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Survodutide

Fat Loss

Phase 2 obesity trial used dose-escalation up to 6 mg/week over 46 weeks. Phase 3 program ongoing for obesity and MASH.

limited human data

Sustanon 250

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Synephrine

Fat Loss

Fat Loss reference profile.

preclinical only· WADA banned

Tabimorelin

GH Secretagogue

GH Secretagogue reference profile.

preclinical only

Tamoxifen

Metabolic

Metabolic reference profile.

preclinical only

Taurine

Metabolic

Metabolic reference profile.

preclinical only

TB-500

Healing

Spreads systemically unlike BPC-157's more localized action

limited human data

Terbutaline

Fat Loss

Fat Loss reference profile.

preclinical only· WADA banned

Tesamorelin

GH Secretagogue

12-16 week minimum for body composition changes. Up to 6 months.

strong human data· WADA banned

Testolactone

Metabolic

Metabolic reference profile.

preclinical only

Testosterone

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Testosterone Cream

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Testosterone Cypionate

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Testosterone Decanoate

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Testosterone Enanthate

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

testosterone furoate

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Testosterone Gel

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Testosterone Isocaproate

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Testosterone Pellets

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Testosterone Phenylpropionate

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Testosterone Propionate

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Testosterone Suspension

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Testosterone Undecanoate

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Tetrahydrogestrinone

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Teverelix

Healing

Healing reference profile.

preclinical only

Theacrine

Fat Loss

Fat Loss reference profile.

preclinical only· WADA banned

Thymalin

Healing

Healing reference profile.

preclinical only

Thymosin Alpha-1

Anti-Inflammatory

Approved in 30+ countries (not US) as Zadaxin for hepatitis B, used adjunctively for hepatitis C and as an oncology adjunct. Twice-weekly…

strong human data

Thymosin Beta-4

Healing

Healing reference profile.

preclinical only

Thymulin

Healing

Healing reference profile.

preclinical only

Tibolone

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Tiomesterone

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Tirzepatide

Metabolic

FDA-approved dual GIP/GLP-1 RA. Start 2.5 mg weekly, increase by 2.5 mg every 4 weeks as tolerated.

strong human data

Toremifene

Metabolic

Metabolic reference profile.

preclinical only

Trenbolone

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Trenbolone Acetate

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Trenbolone Enanthate

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Trenbolone Hexahydrobenzylcarbonate

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Trendione

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Trestolone

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Trestolone Acetate

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Triptorelin

Healing

Healing reference profile.

limited human data

Turinabol

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Urofollitropin

Metabolic

Metabolic reference profile.

preclinical only

Vesugen

Healing

Healing reference profile.

preclinical only

Vilanterol

Fat Loss

Fat Loss reference profile.

preclinical only· WADA banned

Vilon

Healing

Healing reference profile.

preclinical only

Vinyltestosterone

Metabolic

Metabolic reference profile.

preclinical only· WADA banned

Vitamin D3

Metabolic

Metabolic reference profile.

preclinical only

Vorozole

Metabolic

Metabolic reference profile.

preclinical only

YK-11

SARM

Marketed as a SARM but classified as a steroidal myostatin modulator in the literature. No published human trials — dosing is anecdotal.

preclinical only· WADA banned

Yohimbine

Fat Loss

Fat Loss reference profile.

preclinical only· WADA banned

Zinc

Metabolic

Metabolic reference profile.

preclinical only

Zomacton

Healing

Healing reference profile.

preclinical only

zuclomiphene

Metabolic

Metabolic reference profile.

preclinical only

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Reference information only. Always confirm with your clinician before changing your protocol.